Personalized Therapeutics. The Power of Epigenetics.
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Pipeline

Epizyme is leading the creation of small molecule histone methyltransferase inhibitors (HMTi), a new class of personalized therapeutics for the treatment of patients with genetically defined cancers, based on breakthroughs in the field of epigenetics. Genetic alterations in HMTs, a family of epigenetic enzymes, drive multiple human diseases. Our approach represents the future of healthcare by matching better medicines with the right patients.

Our two most advanced therapeutic product programs, targeting the HMTs DOT1L and EZH2, exemplify our approach to creating personalized therapeutics.